January 24
2023
American Society of Clinical Oncology Plenary Series Session
Mutational heterogeneity of imatinib resistance and efficacy of ripretinib vs sunitinib in patients with gastrointestinal stromal tumor: ctDNA analysis from INTRIGUE.
August 10
2022
Journal of Clinical Oncology
Ripretinib Versus Sunitinib in Patients With Advanced Gastrointestinal Stromal Tumor After Treatment With Imatinib (INTRIGUE): A Randomized, Open-Label, Phase III Trial.
June 24
2022
ESMO Open
Efficacy and safety of ripretinib in patients with KIT-altered metastatic melanoma.
May 13
2022
Clinical Pharmacology in Drug Development
Effects of CYP3A Inhibition, CYP3A Induction, and Gastric Acid Reduction on the Pharmacokinetics of Ripretinib, a Switch Control KIT Tyrosine Kinase Inhibitor.
